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Living document · 30 of 44 rows re-verified July 16, 2026

Regulatory Tracker

Peptide regulatory status tracker

Whether a peptide is “legal” is four separate questions with four different answers: is it an FDA-approved drug, may a pharmacy compound it, is it banned in sport, and is it just a research chemical. This table answers all four per compound, and shows the date each row was last checked.

Reviewed by Grey Peptides Editorial Board · ✓ Primary-sourced · Not legal advice

Jul 30
Extended deadline to comment on the GLP-1 503B proposal — FDA-2018-N-3240
7
Peptides before the PCAC on July 23–24 — FDA staff propose adding none
12
Removed from Category 2 in April 2026 — in limbo, not cleared
18
Compounds here named outright on the 2026 WADA Prohibited List
Live · Advisory committee · One week out
PCAC meets July 23–24 on seven peptides — FDA staff propose adding none of them
BPC-157, KPV, TB-500, MOTS-c, emideltide (DSIP), semax and epitalon. All seven nominations were withdrawn; FDA is evaluating anyway. Per-compound briefings, what a vote changes, and what to watch. Docket FDA-2025-N-6895
Compound
Legal path
503A compounding
PCAC review
WADA 2026
Reviewed
BPC-157
Body Protection Compound 157, PL-14736
Legal pathNot FDA-approved
503ALimbo
PCACJul 23, 2026
WADAS0
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 because the nomination was withdrawn — not because FDA cleared it. Not placed on Category 1.
PCAC review
Reviewed for ulcerative colitis. The only one of the seven where FDA cites adverse-event reports involving compounded product. Read the briefing →
WADA 2026 Prohibited List
Named in the 2026 List as an S0 example, on page 4. Prohibited at all times, in and out of competition. S0 substances are Specified Substances.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
BPC-157 →
Row last verified
2026-07-16
KPV
Lys-Pro-Val, α-MSH(11-13)
Legal pathNot FDA-approved
503ALimbo
PCACJul 23, 2026
WADAS0?
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
FDA could not locate information on the use of KPV in humans at all — so no conclusion on safety or effectiveness was possible. Read the briefing →
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
KPV →
Row last verified
2026-07-16
TB-500
Thymosin β4 fragment, Tβ4(17-23)
Legal pathNot FDA-approved
503ALimbo
PCACJul 23, 2026
WADAS2.3
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
Unlike most of the seven, FDA found a lack of historical use in compounding for TB-500 specifically. Read the briefing →
WADA 2026 Prohibited List
Named in the 2026 List under S2.3 growth factors, as “Thymosin-ß4 and its derivatives e.g. TB-500”. Prohibited at all times. S2 substances are non-Specified — a heavier default sanction than the S0 catch-all.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
TB-500 →
Row last verified
2026-07-16
MOTS-c
Mitochondrial ORF of the 12S rRNA type-c
Legal pathNot FDA-approved
503ALimbo
PCACJul 23, 2026
WADAS4.4.1
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
A mitochondrial-derived peptide nominated on the strength of largely preclinical metabolic data. Read the briefing →
WADA 2026 Prohibited List
Named in the 2026 List under S4.4.1 as an AMPK activator — “mitochondrial open reading frame of the 12S rRNA-c (MOTS-c)”, alongside AICAR. Prohibited at all times, non-Specified. Not S2, as is often claimed.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
MOTS-c →
Row last verified
2026-07-16
Emideltide (DSIP)
Delta sleep-inducing peptide
Legal pathNot FDA-approved
503ALimbo
PCACJul 24, 2026
WADAS0?
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
The only one of the seven FDA credits with real historical use in compounding — and staff still propose against it. Historical use alone does not carry a substance. Read the briefing →
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
Emideltide (DSIP) →
Row last verified
2026-07-16
Semax
ACTH(4-7)PGP
Legal pathNot FDA-approved
503ALimbo
PCACJul 24, 2026
WADAS0?
Reviewed07-16
Approved outside the US
Russia — not by FDA. Those are different facts.
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
The only one of the seven where FDA says the evidence demonstrated a lack of effectiveness — plus anticoagulant activity and amphetamine potentiation in animals. Read the briefing →
WADA 2026 Prohibited List
Not named on the 2026 List. S0 turns on having no current approval by any governmental regulatory health authority — and this substance is approved outside the US, so whether S0 catches it is genuinely unsettled. Do not read this row either way: ask Global DRO or your anti-doping organisation.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
Semax →
Row last verified
2026-07-16
Epitalon
Epithalon, Epithalamin, AEDG peptide
Legal pathNot FDA-approved
503ALimbo
PCACJul 24, 2026
WADAS0?
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
FDA spells it “epitalon”; most of the literature spells it “epithalon”. A naming inconsistency FDA treats as part of the characterisation problem. Read the briefing →
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Docket
FDA-2025-N-6895 — linked in Sources below.
Grey Peptides entry
Epitalon →
Row last verified
2026-07-16
GHK-Cu (injectable)
Copper peptide, glycyl-L-histidyl-L-lysine copper
Legal pathNot FDA-approved
503ALimbo
PCACBy Feb 2027
WADAS0?
Reviewed05-19
503A compounding
Removed from Category 2 in April 2026, route-specific — the injectable form. Topical cosmetic use is a separate question this list does not address.
PCAC review
Slated for review by the end of February 2027. No date set.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
GHK-Cu (injectable) →
Row last verified
2026-05-19
Melanotan II
MT-II
Legal pathNot FDA-approved
503ALimbo
PCACBy Feb 2027
WADAS0?
Reviewed05-19
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
Slated for review by the end of February 2027. No date set.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
Melanotan II →
Row last verified
2026-05-19
Cathelicidin (LL-37)
LL-37, hCAP18
Legal pathNot FDA-approved
503ALimbo
PCACBy Feb 2027
WADAS0?
Reviewed05-19
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
Slated for review by the end of February 2027. No date set.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
Cathelicidin (LL-37) →
Row last verified
2026-05-19
Dihexa
N-hexanoic-Tyr-Ile-(6) aminohexanoic amide
Legal pathNot FDA-approved
503ALimbo
PCACBy Feb 2027
WADAS0?
Reviewed05-19
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
Slated for review by the end of February 2027. No date set.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
Dihexa →
Row last verified
2026-05-19
PEG-MGF
Pegylated mechano growth factor
Legal pathNot FDA-approved
503ALimbo
PCACBy Feb 2027
WADAS2.3
Reviewed07-16
503A compounding
Removed from Category 2 in April 2026 (nomination withdrawn). Not placed on Category 1.
PCAC review
Slated for review by the end of February 2027. No date set.
WADA 2026 Prohibited List
The 2026 List names “Mechano growth factors (MGFs)” under S2.3. Prohibited at all times, non-Specified.
Grey Peptides entry
PEG-MGF →
Row last verified
2026-07-16
Semaglutide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed07-16
Brand names
Ozempic, Wegovy, Rybelsus
503A compounding
503A patient-specific compounding can still occur where a prescriber documents a specific clinical need, within FDA's “essentially a copy” limits.
503B bulks list
FDA proposes not to include it on the 503B Bulks List, finding no clinical need. It was never on that list — “removed from” is wrong. Comment period runs to July 30, 2026.
Shortage status
Resolved. The shortage pathway that once permitted compounding is closed.
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Docket
FDA-2018-N-3240 — linked in Sources below.
Grey Peptides entry
Semaglutide →
Row last verified
2026-07-16
Tirzepatide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed07-16
Brand names
Mounjaro, Zepbound
503B bulks list
Same proposal, same docket, same July 30 deadline. Eli Lilly filed comments on tirzepatide; the Outsourcing Facilities Association filed against.
Shortage status
Resolved. The shortage pathway that once permitted compounding is closed.
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Docket
FDA-2018-N-3240 — linked in Sources below.
Grey Peptides entry
Tirzepatide →
Row last verified
2026-07-16
Liraglutide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed07-16
Brand names
Victoza, Saxenda
503B bulks list
Same proposal, same docket, same July 30 deadline.
Shortage status
Resolved. The shortage pathway that once permitted compounding is closed.
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Docket
FDA-2018-N-3240 — linked in Sources below.
Grey Peptides entry
Liraglutide →
Row last verified
2026-07-16
Dulaglutide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed05-19
Brand names
Trulicity
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Grey Peptides entry
Dulaglutide →
Row last verified
2026-05-19
Exenatide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed05-19
Brand names
Byetta, Bydureon
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Grey Peptides entry
Exenatide →
Row last verified
2026-05-19
Orforglipron
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed05-19
Brand names
Foundayo
503A compounding
Approved April 2026. A GLP-1 agonist but a small molecule, not a peptide — it is here because it is constantly miscategorised.
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Grey Peptides entry
Orforglipron →
Row last verified
2026-05-19
Somatropin
Legal pathFDA-approved
503A
PCAC
WADAS2.2.3
Reviewed07-16
Brand names
multiple
WADA 2026 Prohibited List
Growth hormone is named under S2.2.3, with its analogues and fragments. Prohibited at all times, non-Specified. Approval does not exempt a substance from the List.
Grey Peptides entry
Somatropin →
Row last verified
2026-07-16
Teriparatide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed05-19
Brand names
Forteo
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Grey Peptides entry
Teriparatide →
Row last verified
2026-05-19
Octreotide
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed05-19
Brand names
Sandostatin
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Grey Peptides entry
Octreotide →
Row last verified
2026-05-19
Leuprolide
Legal pathFDA-approved
503A
PCAC
WADAS2.2.1
Reviewed07-16
Brand names
Lupron
WADA 2026 Prohibited List
Named as “leuprorelin”, a GnRH agonist analogue under S2.2.1 — prohibited in males only. Prohibited at all times, non-Specified.
Grey Peptides entry
Leuprolide →
Row last verified
2026-07-16
Tesamorelin
Legal pathFDA-approved
503A
PCAC
WADAS2.2.4
Reviewed07-16
Brand names
Egrifta
WADA 2026 Prohibited List
Named under S2.2.4 as a GHRH analogue. FDA-approved and WADA-prohibited at the same time — the two regimes are unrelated.
Grey Peptides entry
Tesamorelin →
Row last verified
2026-07-16
IGF-1 (mecasermin)
Legal pathFDA-approved
503A
PCAC
WADAS2.3
Reviewed07-16
Brand names
Increlex
WADA 2026 Prohibited List
Named under S2.3 as “Insulin-like growth factor 1 (IGF-1, mecasermin) and its analogues”. Prohibited at all times, non-Specified.
Grey Peptides entry
IGF-1 (mecasermin) →
Row last verified
2026-07-16
Bremelanotide (PT-141)
Legal pathFDA-approved
503A
PCAC
WADA
Reviewed05-19
Brand names
Vyleesi
WADA 2026 Prohibited List
Not on the 2026 Prohibited List.
Grey Peptides entry
Bremelanotide (PT-141) →
Row last verified
2026-05-19
SS-31 (elamipretide)
Legal pathFDA-approved
503A
PCAC
WADAS0?
Reviewed07-17
Brand names
Forzinity
503A compounding
Accelerated approval Sept 19, 2025 (Forzinity, NDA 215244) for muscle strength in Barth syndrome at ≥30 kg — the first approved mitochondria-targeted therapeutic. Continued approval contingent on confirmatory trials.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
SS-31 (elamipretide) →
Row last verified
2026-07-17
hCG
Legal pathFDA-approved
503A
PCAC
WADAS2.2.1
Reviewed07-16
Brand names
Pregnyl, Ovidrel
WADA 2026 Prohibited List
Named as “chorionic gonadotrophin (CG)” under S2.2.1 — a testosterone-stimulating peptide, prohibited in males only. Prohibited at all times, non-Specified.
Grey Peptides entry
hCG →
Row last verified
2026-07-16
Retatrutide
Legal pathInvestigational
503A
PCAC
WADAS0?
Reviewed05-19
503A compounding
Not approved anywhere. Not compoundable. Widely sold as a research chemical regardless — see the Retatrutide hub.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
Retatrutide →
Row last verified
2026-05-19
CagriSema
Legal pathInvestigational
503A
PCAC
WADAS0?
Reviewed05-19
503A compounding
Phase 3. A GLP-1 + amylin combination.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
CagriSema →
Row last verified
2026-05-19
Survodutide
Legal pathInvestigational
503A
PCAC
WADAS0?
Reviewed05-19
503A compounding
Phase 3. A GLP-1 + glucagon dual agonist.
WADA 2026 Prohibited List
Not named on the 2026 List. The S0 catch-all covers any substance with no current approval by any governmental regulatory health authority — which, on its face, captures this. Inference, not a WADA ruling: confirm with Global DRO or your anti-doping organisation.
Grey Peptides entry
Survodutide →
Row last verified
2026-05-19
Selank
Legal pathNot FDA-approved
503A
PCAC
WADAS0?
Reviewed07-16
Approved outside the US
Russia — not by FDA. Those are different facts.
503A compounding
Not FDA-approved and not on any US compounding list.
WADA 2026 Prohibited List
Not named on the 2026 List. S0 turns on having no current approval by any governmental regulatory health authority — and this substance is approved outside the US, so whether S0 catches it is genuinely unsettled. Do not read this row either way: ask Global DRO or your anti-doping organisation.
Grey Peptides entry
Selank →
Row last verified
2026-07-16
Noopept
Legal pathNot FDA-approved
503A
PCAC
WADAS0?
Reviewed07-16
Approved outside the US
Russia — not by FDA. Those are different facts.
503A compounding
Not FDA-approved. A dipeptide-derived nootropic, frequently sold in the US as a supplement ingredient it is not lawfully one.
WADA 2026 Prohibited List
Not named on the 2026 List. S0 turns on having no current approval by any governmental regulatory health authority — and this substance is approved outside the US, so whether S0 catches it is genuinely unsettled. Do not read this row either way: ask Global DRO or your anti-doping organisation.
Grey Peptides entry
Noopept →
Row last verified
2026-07-16
Cerebrolysin
Legal pathNot FDA-approved
503A
PCAC
WADAS0?
Reviewed07-16
Approved outside the US
Austria and ~50 other countries — not by FDA. Those are different facts.
503A compounding
Not FDA-approved. A porcine brain-derived peptide preparation.
WADA 2026 Prohibited List
Not named on the 2026 List. S0 turns on having no current approval by any governmental regulatory health authority — and this substance is approved outside the US, so whether S0 catches it is genuinely unsettled. Do not read this row either way: ask Global DRO or your anti-doping organisation.
Grey Peptides entry
Cerebrolysin →
Row last verified
2026-07-16
Thymosin α-1
Legal pathNot FDA-approved
503ACategory 2
PCAC
WADAS0?
Reviewed07-16
Brand names
Zadaxin
Approved outside the US
~35 countries, not the US — not by FDA. Those are different facts.
503A compounding
Not FDA-approved. Placed in 503A Category 2 in 2023 and not among the twelve removed in April 2026.
WADA 2026 Prohibited List
Not named on the 2026 List. S0 turns on having no current approval by any governmental regulatory health authority — and this substance is approved outside the US, so whether S0 catches it is genuinely unsettled. Do not read this row either way: ask Global DRO or your anti-doping organisation.
Grey Peptides entry
Thymosin α-1 →
Row last verified
2026-07-16
Thymopentin
Legal pathNot FDA-approved
503A
PCAC
WADAS0?
Reviewed07-16
Approved outside the US
some countries outside the US — not by FDA. Those are different facts.
503A compounding
Not FDA-approved.
WADA 2026 Prohibited List
Not named on the 2026 List. S0 turns on having no current approval by any governmental regulatory health authority — and this substance is approved outside the US, so whether S0 catches it is genuinely unsettled. Do not read this row either way: ask Global DRO or your anti-doping organisation.
Grey Peptides entry
Thymopentin →
Row last verified
2026-07-16
Pralmorelin (GHRP-2)
Legal pathNot FDA-approved
503A
PCAC
WADAS2.2.4
Reviewed07-16
Approved outside the US
Japan (diagnostic use) — not by FDA. Those are different facts.
503A compounding
Not FDA-approved.
WADA 2026 Prohibited List
Named under S2.2.4 as “GHRP-2 (pralmorelin)”. Prohibited at all times, non-Specified. Being approved in Japan does not lift this — S2 naming is independent of approval status.
Grey Peptides entry
Pralmorelin (GHRP-2) →
Row last verified
2026-07-16
CJC-1295
Legal pathNot FDA-approved
503ACategory 2
PCAC
WADAS2.2.4
Reviewed07-16
503A compounding
Not FDA-approved. Placed in 503A Category 2 in 2023; not among the twelve removed in April 2026.
WADA 2026 Prohibited List
Named under S2.2.4 as a GHRH analogue, alongside CJC-1293. Prohibited at all times, non-Specified.
Grey Peptides entry
CJC-1295 →
Row last verified
2026-07-16
Ipamorelin
Legal pathNot FDA-approved
503ACategory 2
PCAC
WADAS2.2.4
Reviewed07-16
503A compounding
Not FDA-approved. Placed in 503A Category 2 in 2023; not among the twelve removed in April 2026.
WADA 2026 Prohibited List
Named under S2.2.4 as a growth hormone secretagogue. Prohibited at all times, non-Specified.
Grey Peptides entry
Ipamorelin →
Row last verified
2026-07-16
Sermorelin
Legal pathNot FDA-approved
503A
PCAC
WADAS2.2.4
Reviewed07-16
503A compounding
The FDA-approved product (Geref) was discontinued; sermorelin is compounded today rather than dispensed as an approved drug.
WADA 2026 Prohibited List
Named under S2.2.4 as a GHRH analogue. Prohibited at all times, non-Specified.
Grey Peptides entry
Sermorelin →
Row last verified
2026-07-16
GHRP-6
Legal pathNot FDA-approved
503A
PCAC
WADAS2.2.4
Reviewed07-16
503A compounding
Not FDA-approved.
WADA 2026 Prohibited List
Named under S2.2.4 in the GHRP series (GHRP-1 through GHRP-6). Prohibited at all times, non-Specified.
Grey Peptides entry
GHRP-6 →
Row last verified
2026-07-16
Hexarelin
Legal pathNot FDA-approved
503A
PCAC
WADAS2.2.4
Reviewed07-16
503A compounding
Not FDA-approved.
WADA 2026 Prohibited List
Named under S2.2.4 as “examorelin (hexarelin)”. Prohibited at all times, non-Specified.
Grey Peptides entry
Hexarelin →
Row last verified
2026-07-16
MK-677 (ibutamoren)
Legal pathNot FDA-approved
503A
PCAC
WADAS2.2.4
Reviewed07-16
503A compounding
Not FDA-approved. A small-molecule secretagogue, not a peptide — listed here because it is sold and discussed as one.
WADA 2026 Prohibited List
Named under S2.2.4 as “ibutamoren (MK-677)”. Prohibited at all times, non-Specified.
Grey Peptides entry
MK-677 (ibutamoren) →
Row last verified
2026-07-16
AOD-9604
Legal pathNot FDA-approved
503A
PCAC
WADAS2.2.3
Reviewed07-16
503A compounding
Not FDA-approved. Its human obesity trials failed to beat placebo on the primary endpoint — a fact the marketing around it routinely omits.
WADA 2026 Prohibited List
Named under S2.2.3 as a growth hormone fragment, alongside hGH 176-191. Prohibited at all times, non-Specified.
Grey Peptides entry
AOD-9604 →
Row last verified
2026-07-16
Tesofensine
Legal pathNot FDA-approved
503A
PCAC
WADAS6.B
Reviewed07-16
Approved outside the US
Mexico (COFEPRIS) — not by FDA. Those are different facts.
503A compounding
Not FDA-approved. A triple monoamine reuptake inhibitor, not a peptide.
WADA 2026 Prohibited List
Named under S6.B as a Specified Stimulant — prohibited in-competition only, unlike everything else on this page.
Grey Peptides entry
Tesofensine →
Row last verified
2026-07-16

Tap any row for the detail, the reasoning and the docket. Reviewed is the date that row was last checked against a primary source — not the date the page was published. Rows still showing 05-19 were carried forward from the previous review and are flagged as such rather than silently re-dated.

How to read this table

Four independent questions, four columns. Collapsing them is where nearly every wrong answer about peptide legality comes from.

Legal path. FDA-approved means a real prescription medicine with guaranteed identity, dose and sterility. Investigational means it is in trials and not approved anywhere. Not FDA-approved is the largest group, and it includes several compounds that are approved in other countries — which is not the same thing, and is filed separately here for exactly that reason.

503A compounding. Section 503A covers patient-specific compounding by a pharmacy against an individual prescription; section 503B covers outsourcing facilities compounding from bulk. Each keeps its own list. On the 503A interim list, Category 1 means under evaluation with no significant safety concerns identified, and compounding is generally permitted under enforcement discretion. Category 2 means significant safety concerns — not permitted. Category 3 means the nomination lacked enough information to evaluate.

Limbo is not an FDA term. It is this tracker's label for the twelve peptides removed from Category 2 in April 2026 whose nominations had been withdrawn. They were not cleared and they were not moved to Category 1. They are off the do-not-compound list and still not lawful to compound — a state the category system has no name for, which is precisely why it gets misreported as approval.

PCAC review. The Pharmacy Compounding Advisory Committee advises FDA on whether a substance belongs on the 503A Bulks List. It sits on July 23–24, 2026 for the first seven. A recommendation is non-binding, and even a favourable vote must clear notice-and-comment rulemaking that can run past a year. When the committee last looked at peptides in 2024 it recommended against all of them.

WADA 2026. The section of the 2026 WADA Prohibited List that captures the compound. A code in red means the substance is named in the List by name — we read the List to check, rather than repeating what other sites say. A code in amber with a question mark means it is not named and the S0 catch-all is being applied by inference. That distinction is ours, not WADA's, and it exists because the inference is not always safe: S0 only captures substances with no current approval by any governmental health authority, so for a compound registered in Russia or Japan the catch-all may not apply at all. If you are tested, Global DRO and your anti-doping organisation are the answer, not this page.

One asymmetry worth internalising: non-approval can pull a substance onto the WADA list, but approval never pulls one off. Somatropin, tesamorelin, leuprolide, mecasermin and hCG are all FDA-approved and all prohibited at all times. A PCAC vote in July changes nothing about anti-doping status.


The GLP-1 situation, stated accurately

Most coverage says FDA moved to “remove” or “exclude” semaglutide, tirzepatide and liraglutide from the 503B bulks list. That is not what happened, and the error matters.

Those three were never on the 503B Bulks List. They were nominated for it. On May 1, 2026, FDA published a notice — not a final rule — setting out its proposal not to include them, having found no clinical need for outsourcing facilities to compound them from bulk when approved products are available (91 FR 23431, Docket FDA-2018-N-3240). Nothing was delisted, because nothing was listed.

The practical difference is that a proposal is still open. FDA's original comment window closed June 30. After a request for more time, the agency extended it by thirty days, and comments now close July 30, 2026 (91 FR 38719, published June 26). FDA specifically asked that comments address the clinical-need standard in the statute. Trackers still showing a June deadline — including this one until today — are wrong about a window that is currently open.

What has not changed: 503A patient-specific compounding can still occur where a prescriber documents a specific clinical need for an individual patient, within FDA's “essentially a copy” limits. The shortage pathway, which is what actually enabled mass compounding from 2022, closed when FDA declared the semaglutide shortage resolved in February 2025. The direction of travel is toward the approved products.


Change log

What moved, and when. Newest first.

DateChange
2026-07-16Tracker rebuilt as a per-compound table with per-row review dates. WADA column added, verified line by line against the 2026 Prohibited List. Corrected the GLP-1 503B framing from “excluded from” to “proposed not to include”.
2026-06-26FDA extended the 503B GLP-1 comment period by 30 days, to July 30, 2026 (91 FR 38719). The previous version of this tracker still showed the original June deadline.
2026-06-29FDA released briefing documents for all seven PCAC peptides. Staff propose adding none of them.
2026-05-01FDA published its proposal not to include semaglutide, tirzepatide or liraglutide on the 503B Bulks List (91 FR 23431, Docket FDA-2018-N-3240).
2026-04-30FDA announced the 503B GLP-1 proposal.
2026-04-22Twelve peptides formally removed from 503A Category 2 (effective date).
2026-04-15FDA announced the Category 2 removals and scheduled PCAC for July 23-24, 2026.
2026-04-01Orforglipron (Foundayo) approved by FDA.
2025-02FDA declared the semaglutide shortage resolved, beginning the close of GLP-1 compounding.
2023FDA placed 19 peptides into 503A Category 2.

Spot something out of date? This is a living document — email editors@greypeptides.com and we'll verify and update.


Frequently asked questions

Which peptides are FDA approved in 2026?

Approved peptide medicines include semaglutide (Ozempic, Wegovy, Rybelsus), tirzepatide (Mounjaro, Zepbound), liraglutide (Victoza, Saxenda), dulaglutide (Trulicity), exenatide, somatropin, teriparatide, octreotide, leuprolide, tesamorelin (Egrifta), mecasermin (Increlex) and bremelanotide (Vyleesi). Orforglipron (Foundayo, approved April 2026) is a GLP-1 agonist but a small molecule, not a peptide. BPC-157, TB-500, MOTS-c, KPV, semax, epitalon and DSIP are not approved by FDA and are not currently lawful to compound.

Is BPC-157 legal in 2026?

It is not FDA approved and has no USP monograph. In April 2026 it was removed from the 503A Category 2 list because the nomination was withdrawn — not because FDA cleared it — and it was not moved to Category 1, so it is neither flagged nor permitted. FDA's Pharmacy Compounding Advisory Committee reviews it on July 23, 2026, and FDA staff have already proposed not adding it. Separately, BPC-157 is named by name on the 2026 WADA Prohibited List under S0, so it is prohibited at all times for tested athletes.

Did the FDA remove GLP-1s from the 503B bulks list?

No, and this is the most common error in coverage of it. Semaglutide, tirzepatide and liraglutide were never on the 503B Bulks List. They were nominated for it, and on May 1, 2026 FDA published its proposal not to include them, finding no clinical need. Nothing was delisted. The distinction matters because a proposal not to include is still open to comment — through July 30, 2026, under Docket FDA-2018-N-3240.

Does removal from Category 2 mean a peptide is legal to compound now?

No. Removal from Category 2 only lifts the significant-safety-concerns designation. It does not place a substance on the Category 1 list and does not authorise compounding. The twelve peptides removed in April 2026 sit in between: no longer formally flagged, and not permitted either. Reaching the 503A Bulks List requires PCAC review and formal rulemaking, which can take more than a year.

Does a peptide's FDA status affect whether it is banned in sport?

Only in one direction, and not the one people assume. WADA's S0 category captures any substance with no current approval by any governmental regulatory health authority, so non-approval can pull a substance onto the list. But approval never pulls one off: somatropin, tesamorelin, leuprolide, mecasermin and hCG are all FDA-approved and all prohibited. The two regimes are unrelated, and a PCAC vote in July would change nothing about anti-doping status.


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From the News Wire

Seven peptides, one committee, zero staff endorsements → FDA pulls 12 peptides off its "do not compound" list → The FDA just proposed ending mass GLP-1 compounding →

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Sources

Primary documents only. Every WADA cell traces to the 2026 Prohibited List itself; every docket number to the Federal Register notice that carries it. Status reflects each row's own review date and can change.

  1. World Anti-Doping Agency — International Standard: Prohibited List 2026, valid 1 January 2026. Read in full; every WADA cell on this page traces to it.
    View source ↗
  2. Federal Register — List of Bulk Drug Substances for Which There Is a Clinical Need Under Section 503B, 91 FR 23431 (May 1, 2026), Docket FDA-2018-N-3240.
    View source ↗
  3. Federal Register — the same notice, Extension of Comment Period, 91 FR 38719 (June 26, 2026). This is the document that moved the deadline to July 30.
    View source ↗
  4. Regulations.gov — Docket FDA-2025-N-6895, the July 2026 PCAC docket, including the seven briefing documents released June 29, 2026.
    View source ↗
  5. FDA — Interim Policy on Compounding Using Bulk Drug Substances Under Section 503A; 503A interim bulks list (Categories 1-3), updated April 15, 2026.
    View source ↗

Educational only — not legal or medical advice. An advisory-committee recommendation is not a rule, and nothing here describes how to obtain or use any substance. Compounding rules vary by state and by substance. Regulatory status changes frequently; verify against primary sources and a qualified professional before relying on it.